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Raw Material | Cabergoline |
---|---|
Water Retention | No significant impact on water retention |
Hepatotoxicity | Low risk, but liver function monitoring is advised for prolonged use |
Lab Test | Blood prolactin levels |
Also known as | Cabaser, Dostinex |
Blood pressure | May cause hypotension (lower blood pressure) |
Trade name | Dostinex, Cabaser |
Storage conditions | Store at room temperature, protect from light and moisture |
Chemical name | 1-[(6-allylergolin-8ОІ-yl)-carbonyl]-1-[3-(dimethylamino)propyl]-3-ethylurea |
Formula | C26H37N5O2 |
Substance class | Ergoline derivative |
Main action | Dopamine D2 receptor agonist |
Half-life | 63 to 68 hours |
Dosage (medical) | Typically 0.25 mg to 1 mg twice a week for hyperprolactinemia |
Dosage (sports) | Not officially recommended for sports uses, typically around 0.25 mg to 0.5 mg per week when used |
Effects | Decreases prolactin levels, can potentially enhance mood and libido |
Side effects | Nausea, headache, dizziness, orthostatic hypotension, constipation, fatigue, heart valve issues in higher doses |
Use in sports | Primarily used to reduce prolactin-related side effects of anabolic steroids |
Manufacturer | SP Laboratories |
Packing | 20 tabs (0.25mg/tab) |
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